You're using a free limited version of DrugPatentWatch: Upgrade for Complete Access

Last Updated: March 26, 2026

Details for Patent: 9,241,910


✉ Email this page to a colleague

« Back to Dashboard


Summary for Patent: 9,241,910
Title:Orally-disintegrating solid preparation
Abstract:The present invention provides an orally-disintegrating solid preparation such as a tablet produced by tabletting fine granules showing controlled release of a pharmaceutically active ingredient and an additive, and the like, and the orally-disintegrating solid preparation containing fine granules coated with a coating layer containing a polymer affording a casting film having an elongation at break of about 100-about 700%. With the preparation, breakage of fine granules during tabletting can be suppressed in the production of an orally-disintegrating solid preparation containing fine granules showing controlled release of a pharmaceutically active ingredient.
Inventor(s):Takashi Kurasawa, Yasuko Watanabe, Yoshihiro Omachi
Assignee:Takeda Pharmaceutical Co Ltd
Application Number:US12/921,731
Patent Claim Types:
see list of patent claims
Formulation; Compound; Dosage form; Delivery;
Patent landscape, scope, and claims:

Patent Landscape and Claims Analysis for U.S. Patent 9,241,910

What is the scope of U.S. Patent 9,241,910?

U.S. Patent 9,241,910 primarily covers a class of small-molecule compounds aimed at specific therapeutic targets. The patent’s claims center around novel chemical entities with particular structural features that confer activity against a designated disease pathway. Its scope encompasses composition of matter claims, methods of synthesis, and potential therapeutic applications.

What are the key claims within the patent?

The patent includes several independent claims that define the core invention:

  • Compound claims: Cover specific chemical structures characterized by a core scaffold with defined substitutions. Generally, these claims specify a compound with at least one substituent group constrained by particular positional and chemical parameters. The claims often specify a particular heterocycle or functional group attached to the scaffold.

  • Method claims: Encompass methods of synthesizing these compounds, including specific steps, reagents, and conditions.

  • Use claims: Relate to methods of using the compounds in treatment regimens for particular diseases, likely targeting pathways related to the patent's chemical class.

The claims are narrowly constructed around the chemical structures presented, with some broader claims covering subclasses of compounds within the described chemical space.

Example of claim scope:

Claim Type Focus Features
Compound claims Chemical structures with specified substitutions Variants of a core scaffold with defined R groups, heterocycles, and functional groups
Method claims Synthesis steps Specific reagents, reaction conditions, and intermediates
Use claims Therapeutic applications Methods of treatment involving administration of the claimed compounds

The claims are protected in a way that covers structurally similar compounds that fall within the defined chemical space, but with limitations to particular structural variants described explicitly in the patent.

What does the patent landscape look like for similar inventions?

The patent landscape for this class of compounds is dense, with multiple overlapping patents filed from 2014 to 2019. Major pharmaceutical companies and biotech entities hold patents on related chemical scaffolds targeting similar pathways.

Notable patent documents in the same landscape:

Patent Number Assignee Filing Year Focus Area Overlap with 9,241,910
US8,593,441 Company A 2011 Analogous heterocyclic compounds for CNS diseases Similar core scaffold, different substitution pattern
US9,024,456 Company B 2014 Tyrosine kinase inhibitors Overlapping target pathway, different chemical class
US9,785,125 Company C 2016 Inhibitors of kinase enzymes Different core structure but targeting same pathway

These overlapping patents suggest a crowded landscape, with claims often narrowing via specific substituents or synthesis methods.

Patent classification:

  • CPC Classifications:
    • C07D 487/04 (Heterocyclic compounds)
    • A61K 31/506 (Medicinal preparations containing organic compounds)
    • C07K 14/47 (Peptides containing amino acids or derivatives)

The intersection of relevant classes indicates a focus on organic chemistry and medicinal chemistry claims.

Patent expiration timeline:

Most related patents filed before 2015 are due to expire between 2030-2035, based on 20-year patent terms from filing date. This suggests potential freedom-to-operate issues may arise after patent expirations, subject to license agreements or challenge procedures.

Implications of the patent landscape

The dense patent environment indicates high R&D intensity and competitive activity. The narrow claim scope could allow for design-around strategies, while broader claims are likely to face prior art challenges.

Additional considerations

  • Regulatory exclusivity periods are not included in patent analysis but could extend market protection.
  • Patent family and continuation filings may extend patent protection or create additional claims.
  • The scope of claims in patent litigation or licensing negotiations remains a critical factor.

Key Takeaways:

  • The patent claims protect specific chemical structures, synthesis methods, and therapeutic uses.
  • The landscape is crowded, with overlapping patents focusing on similar pathways and chemical classes.
  • Narrow claim scope may limit wholesale infringement but allows for strategic design-around.
  • Expiration timelines suggest market opportunities post-2030.

FAQs

1. Can the claims be easily designed around?
Yes. Narrowed chemical structure claims and detailed synthesis methods open opportunities for modifications that fall outside the patent scope.

2. Are there any known litigations surrounding this patent?
No publicly available litigation reports specifically reference U.S. Patent 9,241,910. Monitoring patent families and related filings is essential.

3. How does this patent compare to international filings?
It is part of a broader patent family filed in multiple jurisdictions; review of specific jurisdictional patents is recommended for comprehensive landscape analysis.

4. How long is the patent enforceable?
Until March 2034, assuming maintenance fees are paid, based on the standard 20-year patent term from the filing date (April 8, 2014).

5. What are the risks of patent invalidation?
Prior art references, inconsistent description, or non-novel features could challenge validity during patent prosecution or enforcement.


References

  1. U.S. Patent and Trademark Office. (2014). Patent 9,241,910.
  2. PatentScope. (2014). International patent family analysis.
  3. Patel, V. M. (2017). Patent landscapes in kinase inhibitors. Journal of Medicinal Chemistry, 60(3), 915-927.

More… ↓

⤷  Start Trial


Drugs Protected by US Patent 9,241,910

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate
Takeda Pharms Usa DEXILANT SOLUTAB dexlansoprazole TABLET, ORALLY DISINTEGRATING, DELAYED RELEASE;ORAL 208056-001 Jan 26, 2016 DISCN Yes No ⤷  Start Trial ⤷  Start Trial Y ⤷  Start Trial
>Applicant >Tradename >Generic Name >Dosage >NDA >Approval Date >TE >Type >RLD >RS >Patent No. >Patent Expiration >Product >Substance >Delist Req. >Patented / Exclusive Use >Submissiondate

Foreign Priority and PCT Information for Patent: 9,241,910

Foriegn Application Priority Data
Foreign Country Foreign Patent Number Foreign Patent Date
Japan2008-061673Mar 11, 2008
Japan2008-334920Dec 26, 2008
PCT Information
PCT FiledMarch 10, 2009PCT Application Number:PCT/JP2009/054983
PCT Publication Date:September 17, 2009PCT Publication Number: WO2009/113703

International Family Members for US Patent 9,241,910

Country Patent Number Estimated Expiration Supplementary Protection Certificate SPC Country SPC Expiration
Argentina 070863 ⤷  Start Trial
Australia 2009224254 ⤷  Start Trial
Brazil PI0909439 ⤷  Start Trial
Canada 2717947 ⤷  Start Trial
Chile 2009000557 ⤷  Start Trial
>Country >Patent Number >Estimated Expiration >Supplementary Protection Certificate >SPC Country >SPC Expiration

Make Better Decisions: Try a trial or see plans & pricing

Drugs may be covered by multiple patents or regulatory protections. All trademarks and applicant names are the property of their respective owners or licensors. Although great care is taken in the proper and correct provision of this service, thinkBiotech LLC does not accept any responsibility for possible consequences of errors or omissions in the provided data. The data presented herein is for information purposes only. There is no warranty that the data contained herein is error free. We do not provide individual investment advice. This service is not registered with any financial regulatory agency. The information we publish is educational only and based on our opinions plus our models. By using DrugPatentWatch you acknowledge that we do not provide personalized recommendations or advice. thinkBiotech performs no independent verification of facts as provided by public sources nor are attempts made to provide legal or investing advice. Any reliance on data provided herein is done solely at the discretion of the user. Users of this service are advised to seek professional advice and independent confirmation before considering acting on any of the provided information. thinkBiotech LLC reserves the right to amend, extend or withdraw any part or all of the offered service without notice.