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Serving leading biopharmaceutical companies globally:

US Army
Healthtrust
Johnson and Johnson
US Department of Justice
Citi
Merck
Chinese Patent Office
Express Scripts
Harvard Business School
Deloitte

Generated: February 22, 2018

DrugPatentWatch Database Preview

Details for Patent: 8,106,183

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Summary for Patent: 8,106,183
Title:Process for preparing an A.sub.2A-adenosine receptor agonist and its polymorphs
Abstract: Disclosed is a synthesis suitable for large scale manufacture of an A.sub.2A-adenosine receptor agonist, and also relates to polymorphs of that compound, and to methods of isolating a specific polymorph.
Inventor(s): Zablocki; Jeff (Mountain View, CA), Elzein; Elfaith (Fremont, CA)
Assignee: Gilead Sciences, Inc. (Foster City, CA)
Application Number:12/765,623
Patent Claim Types:
see list of patent claims
Compound; Use; Process;

Drugs Protected by US Patent 8,106,183

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Patent Submitted
Astellas LEXISCAN regadenoson SOLUTION;INTRAVENOUS 022161-001 Apr 10, 2008 RX Yes Yes ➤ Try a Free Trial ➤ Try a Free Trial Y ➤ Try a Free Trial
Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Patent Submitted

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Non-Orange Book US Patents Family Members for Patent 8,106,183

For Orange Book-listed patents (shown in the main table above) generic applications must certify that the listed patents are expired, invalid, or will not be infringed by generic entry.

The non-Orange Book patents listed below do not require formal certifications, so they do not automatically impede generic entry. Instead, they represent potential opportunities for branded firms to block generic entry through patent infringment challenges.

Patent No. Title Estimated Patent Expiration
7,671,192 Process for preparing an A.sub.2A-adenosine receptor agonist and its polymorphs ➤ Try a Free Trial
8,268,988 Process for preparing an A2A-adenosine receptor agonist and its polymorphs ➤ Try a Free Trial
8,524,883 Monohydrate of (1-{9-[4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-6-aminopu- rin-2-yl}pyrazol-4-yl)-N-methylcarboxamide ➤ Try a Free Trial
9,085,601 Process for preparing an A2A-adenosine receptor agonist and its polymorphs ➤ Try a Free Trial
7,732,595 Process for preparing an A.sub.2A-adenosine receptor agonist and its polymorphs ➤ Try a Free Trial
7,956,179 Process for preparing an A2A-adenosine receptor agonist and its polymorphs ➤ Try a Free Trial
Patent No. Title Estimated Patent Expiration

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International Patents Family Members for US Patent 8,106,183

Country Document Number Estimated Expiration Supplementary Protection Certificate SPC Country SPC Expiration
European Patent Office 1989214 ➤ Try a Free Trial
European Patent Office 2581381 ➤ Try a Free Trial
Spain 2593028 ➤ Try a Free Trial
Israel 193153 ➤ Try a Free Trial
Japan 2009525347 ➤ Try a Free Trial
Japan 5326156 ➤ Try a Free Trial
Japan 2013010791 ➤ Try a Free Trial
South Korea 20080090491 ➤ Try a Free Trial
Japan 2013014620 ➤ Try a Free Trial
South Korea 20130130868 ➤ Try a Free Trial
Country Document Number Estimated Expiration Supplementary Protection Certificate SPC Country SPC Expiration

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Serving hundreds of leading biopharmaceutical companies globally:

Harvard Business School
Mallinckrodt
QuintilesIMS
Daiichi Sankyo
Cipla
Dow
Johnson and Johnson
US Department of Justice
Express Scripts

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