Last Updated: November 13, 2026

Details for Patent: 12,594,243

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Which drugs does patent 12,594,243 protect, and when does it expire?

Patent 12,594,243 protects BRENZAVVY and is included in one NDA.

This patent has twelve patent family members in eleven countries.

Summary for Patent: 12,594,243
Title:Pharmaceutical formulations
Abstract:The pharmacokinetic profile of the SGLT2 inhibitor bexagliflozin can be improved by formulating it as an extended release tablet. Compared with standard immediate-release dosage forms these tablets can permit a lower peak plasma concentration, Cmax, while maintaining plasma concentrations at therapeutic levels for a desired period. This can be used, for instance, to administer lower doses while still providing the same pharmacological effect.
Inventor(s):Feng Wang, Ankit Shrivastava, Rina Shah, Brian Seed, Vinay Patil, Michael J. Hadd, Fuxia DONG, Vipan DHALL, Chunfeng DAI, Joseph Ho-Lun CHAU, Qiuhua CAI
Assignee: Theracosbio LLC
Application Number:US18/501,714
Patent Claim Types:
see list of patent claims
Formulation; Compound; Dosage form;

Drugs Protected by US Patent 12,594,243

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate
Theracosbio BRENZAVVY bexagliflozin TABLET;ORAL 214373-001 Jan 20, 2023 RX Yes Yes ⤷  Start Trial ⤷  Start Trial Y ⤷  Start Trial
>Applicant >Tradename >Generic Name >Dosage >NDA >Approval Date >TE >Type >RLD >RS >Patent No. >Patent Expiration >Product >Substance >Delist Req. >Patented / Exclusive Use >Submissiondate

International Family Members for US Patent 12,594,243

Country Patent Number Estimated Expiration Supplementary Protection Certificate SPC Country SPC Expiration
Argentina 123691 ⤷  Start Trial
Australia 2021357691 ⤷  Start Trial
Canada 3197660 ⤷  Start Trial
China 116600791 ⤷  Start Trial
European Patent Office 4225273 ⤷  Start Trial
>Country >Patent Number >Estimated Expiration >Supplementary Protection Certificate >SPC Country >SPC Expiration

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