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QuintilesIMS
Healthtrust
McKesson
Harvard Business School
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Fish and Richardson
Cipla
Boehringer Ingelheim
Daiichi Sankyo

Generated: May 28, 2018

DrugPatentWatch Database Preview

Crizotinib - Generic Drug Details

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What are the generic drug sources for crizotinib and what is the scope of crizotinib patent protection?

Crizotinib
is the generic ingredient in one branded drug marketed by Pf Prism Cv and is included in one NDA. There are five patents protecting this compound. Additional information is available in the individual branded drug profile pages.

Crizotinib has one hundred and forty-four patent family members in forty-seven countries.

One supplier is listed for this compound.
Summary for crizotinib
International Patents:144
US Patents:5
Tradenames:1
Applicants:1
NDAs:1
Suppliers / Packagers: 1
Bulk Api Vendors: 69
Clinical Trials: 99
Patent Applications: 238
Formulation / Manufacturing:see details
DailyMed Link:crizotinib at DailyMed
Synonyms for crizotinib
(R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-am ine
(R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine
(R)-3-[1-(2,6-Dichloro-3-fluoro-phenyl)-ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)-pyridin-2-ylamine
(R)-crizotinib
2-Pyridinamine, 3-((1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1-(4-piperidinyl)-1H-pyrazol-4-yl)-
2-PYRIDINAMINE, 3-[(1R)-1-(2,6-DICHLORO-3-FLUOROPHENYL)ETHOXY]-5-[1-(4-PIPERIDINYL)-1H-PYRAZOL-4-YL]-
3-((1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1-(4-piperidinyl)-1h-pyrazol-4-yl)pyridin-2-amine
3-(1R)-1-(2,6-Dichloro-3-fluorophenyl)ethoxy-5-1-(4-piperidinyl)-1H-pyrazol-4-yl-2-Pyridinamine
3-[(1r)-1-(2,6-Dichloro-3-Fluorophenyl)ethoxy]-5-(1-Piperidin-4-Yl-1h-Pyrazol-4-Yl)pyridin-2-Amine
3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-[
3-[(1R)-1-(2,6-Dichloro-3-fluorophenyl)ethoxy]-5-[1-(4-piperidinyl)-1H-pyrazol-4-yl]-2-pyridinamine
3-[(1R)-1-(2,6-DICHLORO-3-FLUOROPHENYL)ETHOXY]-5-[1-(4-PIPERIDINYL)-1H-PYRAZOL-4-YL]PYRIDIN-2-AMINE
3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-[1-(piperidin-4-yl)-1H-pyrazol-4-yl]pyridin-2-amine
3-[(R)-1-(2,6-Dichloro-3-fluoro-phenyl)-ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)-pyridin-2-ylamine
399P525
53AH36668S
877399-52-5
877399-52-5, 877399-53-6 (acetate)
912279-98-2
AB0027203
ABP000131
AK172044
AKOS015901233
AKOS015995207
AMX10152
ANW-47749
AOB2688
BB 0261738
BC622990
BCPP000116
BDBM50306682
BRD-K78431006-001-01-1
C21H22Cl2FN5O
CHEBI:64310
CHEMBL601719
Crizotinib (JAN/USAN/INN)
Crizotinib (PF-02341066)
Crizotinib (PF-2341066)
Crizotinib [USAN:INN]
Crizotinib, >=98% (HPLC)
crizotinibum
CTK5F8952
D03ZBT
D09731
DB08865
EN002685
EX-A096
FT-0665224
GS-6178
GTPL4903
HY-50878
I14-14837
J-510370
KB-26391
KIN0000318
KS-0000075X
KTEIFNKAUNYNJU-GFCCVEGCSA-N
MFCD12407409
MolPort-009-679-404
NCGC00250400-01
novel ALK inhibitors
NSC-749005
NSC749005
PB11015
PF 02341066
PF 2341066
PF 2341066;(R)-3-[1-(2,6-Dichloro-3-fluoro-phenyl)-ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)-pyridin-2-ylamine
PF-02341066
PF-02341066 (Crizotinib)
PF-2341066
PF-2341066 - Crizotinib
PF-2341066 (Crizotinib)
PF-2341066,Crizotinib
PF-2341066(Crizotinib)
PF2341066
PubChem19322
Q-3209
QCR-32
RL05464
SC-48062
SCHEMBL93829
SYN1139
TX-017903
UNII-53AH36668S
VGH
W9013
Xalkori
Xalkori (TN)
ZINC35902489

US Patents and Regulatory Information for crizotinib

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Exclusivity Expiration
Pf Prism Cv XALKORI crizotinib CAPSULE;ORAL 202570-002 Aug 26, 2011 RX Yes Yes ➤ Sign Up ➤ Sign Up Y Y ➤ Sign Up
Pf Prism Cv XALKORI crizotinib CAPSULE;ORAL 202570-002 Aug 26, 2011 RX Yes Yes ➤ Sign Up ➤ Sign Up ➤ Sign Up
Pf Prism Cv XALKORI crizotinib CAPSULE;ORAL 202570-001 Aug 26, 2011 RX Yes No ➤ Sign Up ➤ Sign Up ➤ Sign Up
Pf Prism Cv XALKORI crizotinib CAPSULE;ORAL 202570-002 Aug 26, 2011 RX Yes Yes ➤ Sign Up ➤ Sign Up ➤ Sign Up
Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Exclusivity Expiration

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Non-Orange Book US Patents for crizotinib

For Orange Book-listed patents (shown in the main table above) generic applications must certify that the listed patents are expired, invalid, or will not be infringed by generic entry.

The non-Orange Book patents listed below do not require formal certifications, so they do not automatically impede generic entry. Instead, they represent potential opportunities for branded firms to block generic entry through patent infringment challenges.

Patent No. Title Estimated Patent Expiration
8,106,197 Aminoheteroaryl compounds as protein kinase inhibitors ➤ Sign Up
Patent No. Title Estimated Patent Expiration

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Supplementary Protection Certificates for crizotinib

Supplementary Protection Certificate SPC Country SPC Expiration SPC Description
9 Finland ➤ Sign Up
13/009 Ireland ➤ Sign Up PRODUCT NAME: PRODUCT (I.E. ACTIVE INGREDIENT OR COMBINATION OF ACTIVE INGREDIENTS) FOR WHICH A CERTIFICATE IS REQUESTED: CRIZOTINIB, OPTIONALLY IN THE FORM OF A PHARMACEUTICALLY ACCEPTABLE SALT, HYDRATE OR SOLVATE THEREOF; REGISTRATION NO/DATE: EU/1/12/793/001 EU/1/12/793/004 20121023
2013005,C1786785 Lithuania ➤ Sign Up PRODUCT NAME: CRIZOTINIBUM; REGISTRATION NO/DATE: EU/1/12/793/001 - EU/1/12/793/004, 0121023
90008-9 Sweden ➤ Sign Up PRODUCT NAME: CRIZOTINIB INKLUSIVE ETT FARMACEUTISKT GODTAGBART SALT, SOLVAT ELLER HYDRAT DAERAV; REG. NO/DATE: EU/1/12/793/001 20121023
Supplementary Protection Certificate SPC Country SPC Expiration SPC Description

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Serving hundreds of leading biopharmaceutical companies globally:

Dow
Covington
Fuji
Accenture
UBS
Merck
McKinsey
US Army
Express Scripts

Drugs may be covered by multiple patents or regulatory protections. All trademarks and applicant names are the property of their respective owners or licensors. Although great care is taken in the proper and correct provision of this service, thinkBiotech LLC does not accept any responsibility for possible consequences of errors or omissions in the provided data. The data presented herein is for information purposes only. There is no warranty that the data contained herein is error free. thinkBiotech performs no independent verifification of facts as provided by public sources nor are attempts made to provide legal or investing advice. Any reliance on data provided herein is done solely at the discretion of the user. Users of this service are advised to seek professional advice and independent confirmation before considering acting on any of the provided information. thinkBiotech LLC reserves the right to amend, extend or withdraw any part or all of the offered service without notice.