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Last Updated: December 2, 2021

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Details for Patent: 8,969,336

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Which drugs does patent 8,969,336 protect, and when does it expire?

Patent 8,969,336 protects XOSPATA and is included in one NDA.

This patent has forty-seven patent family members in twenty-eight countries.

Summary for Patent: 8,969,336
Title:Diamino heterocyclic carboxamide compound
Abstract: Provided is a compound useful as an inhibitor against the kinase activity of EML4-ALK fusion protein. As a result of intensive and extensive studies on compounds having inhibitory activity against the kinase activity of EML4-ALK fusion protein, the present inventors found that the diamino heterocyclic carboxamide compounds of the present invention had inhibitory activity against the kinase activity of EML4-ALK fusion protein. By this finding, the present invention was completed. The compounds of the present invention can be used as a pharmaceutical composition for preventing and/or treating cancer, such as lung cancer, non-small cell lung cancer, and small cell lung cancer.
Inventor(s): Shimada; Itsuro (Tokyo, JP), Kurosawa; Kazuo (Tokyo, JP), Matsuya; Takahiro (Tokyo, JP), Iikubo; Kazuhiko (Tokyo, JP), Kondoh; Yutaka (Tokyo, JP), Kamikawa; Akio (Tokyo, JP), Tomiyama; Hiroshi (Nagano, JP), Iwai; Yoshinori (Nagano, JP)
Assignee: Astellas Pharma Inc. (Tokyo, JP) Kotobuki Pharmaceutical Co., Ltd. (Hanishina-gun, JP)
Application Number:13/266,164
Patent Claim Types:
see list of patent claims
Use; Composition; Compound;

Drugs Protected by US Patent 8,969,336

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate
Astellas XOSPATA gilteritinib fumarate TABLET;ORAL 211349-001 Nov 28, 2018 RX Yes Yes ⤷  Free Forever Trial ⤷  Free Forever Trial Y Y ⤷  Free Forever Trial
>Applicant >Tradename >Generic Name >Dosage >NDA >Approval Date >TE >Type >RLD >RS >Patent No. >Patent Expiration >Product >Substance >Delist Req. >Patented / Exclusive Use >Submissiondate

Foreign Priority and PCT Information for Patent: 8,969,336

Foriegn Application Priority Data
Foreign Country Foreign Patent Number Foreign Patent Date
Japan2009-113936May 8, 2009
PCT Information
PCT FiledMay 06, 2010PCT Application Number:PCT/JP2010/057751
PCT Publication Date:November 11, 2010PCT Publication Number: WO2010/128659

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Boehringer Ingelheim

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