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Serving leading biopharmaceutical companies globally:

McKesson
US Army
Moodys
Healthtrust
Argus Health
Covington
Baxter
Fuji
Harvard Business School
Boehringer Ingelheim

Generated: February 24, 2018

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Title:Cyclic peptide antifungal agents and process for preparation thereof
Abstract: Provided are compounds of the formula (1): ##STR00001## wherein R' is hydrogen, methyl or NH.sub.2C(O)CH.sub.2--; R'' and R''' are independently methyl or hydrogen; R adn R.sup.y are independently hydroxy or hydrogen; R.sub.1 is hydroxy, hydrogen, or hydroxysulfonyloxy; R.sub.7 is hydroxy, hydrogen, hydroxysulfonyloxy or phosphonooxy; R.sub.2 is a novel acyl side chain. Also provided are novel formulations, methods of inhibiting fungal and parasitic activity, and a process for preparing dideoxy (R.dbd.H) forms of the compounds.
Inventor(s): Burkhardt; Frederick J. (Indianapolis, IN), Debono; Manuel (Indianapolis, IN), Nissen; Jeffrey S. (Indianapolis, IN), Turner, Jr.; William Wilson (Bloomington, IN)
Assignee: Eli Lilly and Company (Indianapolis, IN)
Filing Date:Mar 10, 2005
Application Number:11/078,791
Claims:1. A pharmaceutical formulation comprising a compound having the following formula: ##STR00237## wherein R is --O(CH.sub.2).sub.3CH.sub.3, --O(CH.sub.2).sub.4CH.sub.3, --O(CH.sub.2).sub.5CH.sub.3, --O(CH.sub.2).sub.2O(CH.sub.2).sub.3CH.sub.3, or --O(CH.sub.2).sub.2OC(CH--.sub.3).sub.3, and a pharmaceutically acceptable carrier, wherein the formulation is formulated for inhalation.

2. The pharmaceutical formulation of claim 1, wherein the formulation comprises an aerosol spray.
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Serving leading biopharmaceutical companies globally:

McKesson
Dow
Harvard Business School
Cipla
Farmers Insurance
Healthtrust
Johnson and Johnson
QuintilesIMS
Julphar
Novartis

Drugs may be covered by multiple patents or regulatory protections. All trademarks and applicant names are the property of their respective owners or licensors. Although great care is taken in the proper and correct provision of this service, thinkBiotech LLC does not accept any responsibility for possible consequences of errors or omissions in the provided data. The data presented herein is for information purposes only. There is no warranty that the data contained herein is error free. thinkBiotech performs no independent verifification of facts as provided by public sources nor are attempts made to provide legal or investing advice. Any reliance on data provided herein is done solely at the discretion of the user. Users of this service are advised to seek professional advice and independent confirmation before considering acting on any of the provided information. thinkBiotech LLC reserves the right to amend, extend or withdraw any part or all of the offered service without notice.

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