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Serving leading biopharmaceutical companies globally:

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Generated: January 23, 2018

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Title: Compounds
Abstract:The invention provides new triazolo[4,5-d]pyrimidine compounds, their use as medicaments, compositions containing them and processes for their preparation.
Inventor(s): Hardern; David (Sutton Bonington, GB), Ingall; Anthony (Loughborough, GB), Springthorpe; Brian (Loughborough, GB), Willis; Paul (West Bridgford, GB), Guile; Simon (Loughborough, GB)
Assignee: AstraZeneca AB (Sodertalje, SE)
Filing Date:Dec 20, 2002
Application Number:10/323,655
Claims:1. A compound of formula (II): ##STR14##

where R.sup.1 is C.sub.3-5 alkyl optionally substituted by 1 or more halogen atoms; R.sup.3 and R.sup.4 are both hydroxy; R is XOH, where X is OCH.sub.2 CH.sub.2, or a protected derivative thereof, or R.sup.3 and R.sup.4 together form a bond in the 5-membered ring, or R is CH.sub.2 CH.sub.2 OR' where R' is C.sub.1-6 alkyl or benzyl, and L is halogen or SR, or said hydroxy groups R.sup.3 and R.sup.4 are protected as groups OP.sup.1 and OP.sup.2 where P.sup.1 and P.sup.2 are protecting groups selected from the group consisting of C.sub.1-6 alkyl, benzyl, (C.sub.1-6 alkyl).sub.3 Si and C(O)C.sub.1-6 alkyl or said groups P.sup.1 and P.sup.2, together with the atoms to which they are attached, may form an alkylidene ring or an alkoxymethylidene ring.

2. A compound of formula (II): ##STR15##

where R.sup.1 is n-propyl; R.sup.3 and R.sup.4 are both hydroxyl; R is OCH.sub.2 CH.sub.2 OH or a protected derivative thereof; and L is halogen or SR, or said hydroxyl groups R.sup.3 and R.sup.4 are protected as groups OP.sup.1 and OP.sup.2 where P.sup.1 and P.sup.2 are protecting groups selected from the group consisting of C.sub.1-6 alkyl, benzyl, C.sub.1-6 alkyl).sub.3 Si and C(O)C.sub.1-6 alkyl or said groups P.sup.1 and P.sup.2, together with the atoms to which they are attached, may form an alkylidene ring or an alkoxymethylidene ring.
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US Department of Justice

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