List of Excipients in API tolvaptan
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Excipients in NDA-approved (novel) drugs containing tolvaptan
| Company | Tradename | Ingredient | NDC | Excipient | Potential Generic Entry |
|---|---|---|---|---|---|
| Otsuka America Pharmaceutical Inc | SAMSCA | tolvaptan | 59148-020 | CELLULOSE, MICROCRYSTALLINE | |
| Otsuka America Pharmaceutical Inc | SAMSCA | tolvaptan | 59148-020 | FD&C BLUE NO. 2--ALUMINUM LAKE | |
| Otsuka America Pharmaceutical Inc | SAMSCA | tolvaptan | 59148-020 | HYDROXYPROPYL CELLULOSE | |
| Otsuka America Pharmaceutical Inc | SAMSCA | tolvaptan | 59148-020 | LACTOSE MONOHYDRATE | |
| Otsuka America Pharmaceutical Inc | SAMSCA | tolvaptan | 59148-020 | LOW-SUBSTITUTED HYDROXYPROPYL CELLULOSE | |
| Otsuka America Pharmaceutical Inc | SAMSCA | tolvaptan | 59148-020 | MAGNESIUM STEARATE | |
| Otsuka America Pharmaceutical Inc | SAMSCA | tolvaptan | 59148-020 | STARCH, CORN | |
| >Company | >Tradename | >Ingredient | >NDC | >Excipient | >Potential Generic Entry |
Excipients in ANDA-approved (generic) drugs containing tolvaptan
Detailed excipient profiles for tolvaptan
Excipient focus: ANHYDROUS LACTOSE
tolvaptan drug variants containing ANHYDROUS LACTOSE
| Company | Ingredient | NDC |
|---|---|---|
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing ANHYDROUS LACTOSE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: CELLULOSE, MICROCRYSTALLINE
tolvaptan drug variants containing CELLULOSE, MICROCRYSTALLINE
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing CELLULOSE, MICROCRYSTALLINE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: COPOVIDONE K25-31
tolvaptan drug variants containing COPOVIDONE K25-31
| Company | Ingredient | NDC |
|---|---|---|
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing COPOVIDONE K25-31
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: CROSCARMELLOSE SODIUM
tolvaptan drug variants containing CROSCARMELLOSE SODIUM
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing CROSCARMELLOSE SODIUM
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| >Company | >Ingredient | >NDC |
Excipient focus: FD&C BLUE NO. 2
tolvaptan drug variants containing FD&C BLUE NO. 2
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing FD&C BLUE NO. 2
| Company | Ingredient | NDC |
|---|---|---|
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: FD&C BLUE NO. 2 ALUMINUM LAKE
tolvaptan drug variants containing FD&C BLUE NO. 2 ALUMINUM LAKE
| Company | Ingredient | NDC |
|---|---|---|
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing FD&C BLUE NO. 2 ALUMINUM LAKE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| >Company | >Ingredient | >NDC |
Excipient focus: FD&C BLUE NO. 2--ALUMINUM LAKE
tolvaptan drug variants containing FD&C BLUE NO. 2--ALUMINUM LAKE
| Company | Ingredient | NDC |
|---|---|---|
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing FD&C BLUE NO. 2--ALUMINUM LAKE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: HYDROXYPROPYL CELLULOSE
tolvaptan drug variants containing HYDROXYPROPYL CELLULOSE
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing HYDROXYPROPYL CELLULOSE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| >Company | >Ingredient | >NDC |
Excipient focus: HYDROXYPROPYL CELLULOSE, LOW SUBSTITUTED
tolvaptan drug variants containing HYDROXYPROPYL CELLULOSE, LOW SUBSTITUTED
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing HYDROXYPROPYL CELLULOSE, LOW SUBSTITUTED
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: HYPROMELLOSE 2910
tolvaptan drug variants containing HYPROMELLOSE 2910
| Company | Ingredient | NDC |
|---|---|---|
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing HYPROMELLOSE 2910
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: LACTOSE MONOHYDRATE
tolvaptan drug variants containing LACTOSE MONOHYDRATE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing LACTOSE MONOHYDRATE
| Company | Ingredient | NDC |
|---|---|---|
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| >Company | >Ingredient | >NDC |
Excipient focus: LOW-SUBSTITUTED HYDROXYPROPYL CELLULOSE
tolvaptan drug variants containing LOW-SUBSTITUTED HYDROXYPROPYL CELLULOSE
| Company | Ingredient | NDC |
|---|---|---|
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing LOW-SUBSTITUTED HYDROXYPROPYL CELLULOSE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: MAGNESIUM STEARATE
tolvaptan drug variants containing MAGNESIUM STEARATE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing MAGNESIUM STEARATE
| Company | Ingredient | NDC |
|---|---|---|
| >Company | >Ingredient | >NDC |
Excipient focus: METHYL ALCOHOL
tolvaptan drug variants containing METHYL ALCOHOL
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing METHYL ALCOHOL
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: METHYLENE CHLORIDE
tolvaptan drug variants containing METHYLENE CHLORIDE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing METHYLENE CHLORIDE
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: MICROCRYSTALLINE CELLULOSE 102
tolvaptan drug variants containing MICROCRYSTALLINE CELLULOSE 102
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing MICROCRYSTALLINE CELLULOSE 102
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| >Company | >Ingredient | >NDC |
Excipient focus: POVIDONE K30
tolvaptan drug variants containing POVIDONE K30
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing POVIDONE K30
| Company | Ingredient | NDC |
|---|---|---|
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: SILICON DIOXIDE
tolvaptan drug variants containing SILICON DIOXIDE
| Company | Ingredient | NDC |
|---|---|---|
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing SILICON DIOXIDE
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
Excipient focus: STARCH, CORN
tolvaptan drug variants containing STARCH, CORN
| Company | Ingredient | NDC |
|---|---|---|
| Camber Pharmaceuticals Inc | tolvaptan | 31722-869 |
| Endo USA Inc | tolvaptan | 49884-768 |
| Otsuka America Pharmaceutical Inc | tolvaptan | 59148-020 |
| Apotex Corp | tolvaptan | 60505-4704 |
| Ascend Laboratories LLC | tolvaptan | 67877-636 |
| Novadoz Pharmaceuticals LLC | tolvaptan | 72205-130 |
| >Company | >Ingredient | >NDC |
tolvaptan drug variants not containing STARCH, CORN
| Company | Ingredient | NDC |
|---|---|---|
| Apotex Corp | tolvaptan | 60505-4317 |
| Apotex Corp | tolvaptan | 60505-4318 |
| >Company | >Ingredient | >NDC |
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