Details for Patent: 5,965,525
Summary for Patent: 5,965,525
| Title: | Cyclic peptide antifungal agents |
| Abstract: | Provided are compounds of the formula (1): ##STR1## wherein R' is hydrogen, methyl or NH2 C(O)CH2 --;R" and R'" are independently methyl or hydrogen;R and Ry are independently hydroxy or hydrogen;R1 is hydroxy, hydrogen, or hydroxysulfonyloxy;R7 is hydroxy, hydrogen, hydroxysulfonyloxy or phosphonooxy;R2 is a novel acyl side chain. Also provided are novel formulations, methods of inhibiting fungal and parasitic activity, and a process for preparing dideoxy (R=H) forms of the compounds. |
| Inventor(s): | Frederick J. Burkhardt, Manuel Debono, Jeffrey S. Nissen, William W. Turner, Jr. |
| Assignee: | Eli Lilly and Co |
| Application Number: | US08/449,056 |
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Patent Claim Types: see list of patent claims | Use; Composition; Formulation; |
Drugs Protected by US Patent 5,965,525
| Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Submissiondate |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| >Applicant | >Tradename | >Generic Name | >Dosage | >NDA | >Approval Date | >TE | >Type | >RLD | >RS | >Patent No. | >Patent Expiration | >Product | >Substance | >Delist Req. | >Patented / Exclusive Use | >Submissiondate |
International Family Members for US Patent 5,965,525
| Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
|---|---|---|---|---|---|
| European Patent Office | 0561639 | ⤷ Start Trial | 91406 | Luxembourg | ⤷ Start Trial |
| European Patent Office | 0561639 | ⤷ Start Trial | CA 2008 00017 | Denmark | ⤷ Start Trial |
| European Patent Office | 0561639 | ⤷ Start Trial | 300334 | Netherlands | ⤷ Start Trial |
| >Country | >Patent Number | >Estimated Expiration | >Supplementary Protection Certificate | >SPC Country | >SPC Expiration |
