Details for Patent: 5,387,603
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Summary for Patent: 5,387,603
Title: | 1,5,7-trisubstituted indoline compounds and salts thereof |
Abstract: | Indoline compounds represented by the formula: ##STR1## wherein R represents a saturated or unsaturated aliphatic acyl group which may have one or more halogen atoms, a hydroxy group, a lower alkoxy group, a carboxy group, a lower alkoxycarbonyl group, a cycloalkyl group or an aryl group as substituents; a hydroxyalkyl group; an aliphatic acyloxyalkyl group; a lower alkyl group having a lower alkoxy group, a carboxy group, a lower alkoxycarbonyl group, an aryl substituted lower alkoxycarbonyl group, a carbamoyl group, a mono- or dialkyl substituted carbamoyl group or a cyano group as substituents; an aromatic acyl group which may have one or more halogen atoms as substituents; a furoyl group or a pyridylcarbonyl group; R.sup.1 represents a lower alkyl group which may have one or more halogen atoms or an aryl group as substituents; and pharmaceutically acceptable salts thereof, exhibit a selective suppressive action on urethral contractions, and thus are useful as therapeutic agents for the treatment of dysuria with less hypotension including postural hypotension. |
Inventor(s): | Kitazawa; Makio (Nagano, JP), Ban; Masaaki (Nagano, JP), Okazaki; Kosuke (Nagano, JP), Ozawa; Motoyasu (Nagano, JP), Yazaki; Toshikazu (Nagano, JP), Yamagishi; Ryoichi (Nagano, JP) |
Assignee: | Kissei Pharmaceutical Co., Ltd. (Nagano, JP) |
Application Number: | 08/159,624 |
Patent Claim Types: see list of patent claims | Compound; Use; Composition; |
Drugs Protected by US Patent 5,387,603
Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Submissiondate |
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>Applicant | >Tradename | >Generic Name | >Dosage | >NDA | >Approval Date | >TE | >Type | >RLD | >RS | >Patent No. | >Patent Expiration | >Product | >Substance | >Delist Req. | >Patented / Exclusive Use | >Submissiondate |
Foreign Priority and PCT Information for Patent: 5,387,603
Foriegn Application Priority Data | ||
Foreign Country | Foreign Patent Number | Foreign Patent Date |
Japan | 4-356197 | Dec 02, 1992 |
International Family Members for US Patent 5,387,603
Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
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Canada | 2110454 | ⤷ Try a Trial | |||
Germany | 122010000031 | ⤷ Try a Trial | |||
Germany | 69319551 | ⤷ Try a Trial | |||
European Patent Office | 0600675 | ⤷ Try a Trial | C300454 | Netherlands | ⤷ Try a Trial |
European Patent Office | 0600675 | ⤷ Try a Trial | 1090028-0.L | Sweden | ⤷ Try a Trial |
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