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Claims for Patent: 5,021,458

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Claims for Patent: 5,021,458

Title: Amine derivatives and fungicides containing the same
Abstract:Amine derivatives having the general formula (I): ##STR1## wherein X is selected from the group consisting of ##STR2## wherein Q is oxygen, sulfur or nitrogen atom, and ##STR3## wherein Q is as above; Y is selected from the group consisting of ##STR4## R.sup.1 is hydrogen atom or an alkyl group; R.sup.2 is hydrogen atom or an alkyl group; R.sup.3 is hydrogen atom, a halogen atom or an alkyl group; R.sup.4 is hydrogen atom, an alkyl group, a cycloalkyl group, a halogenated alkyl group or a halogen atom; R.sup.5 is hydrogen atom, an alkyl group, an alkoxy group, a halogen atom, nitro group or hydroxy group; R.sup.5 is attached to an arbitrary position of X, and R.sup.3 or R.sup.4 is attached to an arbitrary position of Y. The amine derivatives (I) are useful as fungicides.
Inventor(s): Maeda; Tetsuya (Tokorozawa, JP), Yamamoto; Toshiyuki (Tokyo, JP), Takase; Mituo (Hino, JP), Sasaki; Kazuya (Higashikurume, JP), Arika; Tadashi (Kasukabe, JP), Yokoo; Mamoru (Kawagoe, JP), Hashimoto; Rieko (Asaka, JP), Amemiya; Kouji (Kodaira, JP), Koshikawa; Sakae (Kawaguchi, JP)
Assignee: Kaken Pharmaceutical Co., Ltd. (Tokyo, JP)
Application Number:07/283,055
Patent Claims: 1. Amine derivatives having the formula (I): ##STR100## wherein X is ##STR101## Y is ##STR102## R.sup.1 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R.sup.2 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;

R.sup.3 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;

R.sup.4 is an alkyl group of 1 to 10 carbon atoms, a cycloalkyl group of 3 to 7 atoms or a halogenated alkyl group; R.sup.5 is hydrogen atom, an alkyl group of 1 to 6 carbon atoms, a halogen atom or a nitro group; R.sup.5 is attached to an arbitrary position of X, and R.sup.3 or R.sup.4 is attached to an arbitrary position of Y.

2. Fungicides containing amine derivatives having the formula (I): ##STR103## wherein X is ##STR104## Y is ##STR105## R.sup.1 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R.sup.2 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;

R.sup.3 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;

R.sup.4 is an alkyl group of 1 to 6 carbon atoms, a cycloalkyl group of 3 to 7 carbon atoms or a halogenated alkyl group; R.sup.5 is hydrogen atom, an alkyl group of 1 to 6 carbon atoms, a halogen atom or a nitro group; R.sup.5 is attached to an arbitrary position of X, and R.sup.3 or R.sup.4 is attached to an arbitrary position of Y.

3. A method of controlling fungi in an animal subject, which comprises treating the animal subject with an amine derivative represented by the Formula (I): ##STR106## wherein X is ##STR107## Y is ##STR108## R.sup.1 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R.sup.2 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;

R.sup.3 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;

R.sup.4 is an alkyl group of 1 to 10 carbon atoms, a cycloalkyl group of 3 to 7 carbon atoms or a halogenated alkyl group; R.sup.5 is hydrogen atom, an alkyl group of 1 to 6 carbon atoms, a halogen atom or a nitro group; R.sup.5 is attached to an arbitrary position of X, and R.sup.3 or R.sup.4 is attached to an arbitrary position of Y.
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