Last Updated: May 11, 2026

Claims for Patent: 5,021,458

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Summary for Patent: 5,021,458

Title:	Amine derivatives and fungicides containing the same
Abstract:	Amine derivatives having the general formula (I): (I) wherein X is selected from the group consisting of wherein Q is oxygen, sulfur or nitrogen atom, and wherein Q is as above; Y is selected from the group consisting of R1 is hydrogen atom or an alkyl group; R2 is hydrogen atom or an alkyl group; R3 is hydrogen atom, a halogen atom or an alkyl group; R4 is hydrogen atom, an alkyl group, a cycloalkyl group, a halogenated alkyl group or a halogen atom; R5 is hydrogen atom, an alkyl group, an alkoxy group, a halogen atom, nitro group or hydroxy group; R5 is attached to an arbitrary position of X, and R3 or R4 is attached to an arbitrary position of Y. The amine derivatives (I) are useful as fungicides.
Inventor(s):	Tetsuya Maeda, Toshiyuki Yamamoto, Mituo Takase, Kazuya Sasaki, Tadashi Arika, Mamoru Yokoo, Rieko Hashimoto, Kouji Amemiya, Sakae Koshikawa
Assignee:	Kaken Pharmaceutical Co Ltd
Application Number:	US07/283,055
Patent Claims:	1. Amine derivatives having the formula (I): ##STR100## wherein X is ##STR101## Y is ##STR102## R1 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R2 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;R3 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R4 is an alkyl group of 1 to 10 carbon atoms, a cycloalkyl group of 3 to 7 atoms or a halogenated alkyl group; R5 is hydrogen atom, an alkyl group of 1 to 6 carbon atoms, a halogen atom or a nitro group; R5 is attached to an arbitrary position of X, and R3 or R4 is attached to an arbitrary position of Y. 2. Fungicides containing amine derivatives having the formula (I): ##STR103## wherein X is ##STR104## Y is ##STR105## R1 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R2 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;R3 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R4 is an alkyl group of 1 to 6 carbon atoms, a cycloalkyl group of 3 to 7 carbon atoms or a halogenated alkyl group; R5 is hydrogen atom, an alkyl group of 1 to 6 carbon atoms, a halogen atom or a nitro group; R5 is attached to an arbitrary position of X, and R3 or R4 is attached to an arbitrary position of Y. 3. A method of controlling fungi in an animal subject, which comprises treating the animal subject with an amine derivative represented by the Formula (I): ##STR106## wherein X is ##STR107## Y is ##STR108## R1 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R2 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms;R3 is hydrogen atom or an alkyl group of 1 to 6 carbon atoms; R4 is an alkyl group of 1 to 10 carbon atoms, a cycloalkyl group of 3 to 7 carbon atoms or a halogenated alkyl group; R5 is hydrogen atom, an alkyl group of 1 to 6 carbon atoms, a halogen atom or a nitro group; R5 is attached to an arbitrary position of X, and R3 or R4 is attached to an arbitrary position of Y.

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