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Last Updated: September 26, 2020

DrugPatentWatch Database Preview

Details for Patent: 9,481,663

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Which drugs does patent 9,481,663 protect, and when does it expire?

Patent 9,481,663 protects ERLEADA and is included in one NDA.

This patent has sixty-six patent family members in thirty-seven countries.

Summary for Patent: 9,481,663
Title:Crystalline forms of an androgen receptor modulator
Abstract: Described herein are amorphous and crystalline forms of the androgen receptor modulator 4-[7-(6-cyano-5-trifluoromethylpyridin-3-yl)-8-oxo-6-thioxo-5,7-diazaspir- o[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide. Also described are pharmaceutical compositions suitable for administration to a mammal that include the androgen receptor modulator, and methods of using the androgen receptor modulator, alone and in combination with other compounds, for treating diseases or conditions that are associated with androgen receptor activity.
Inventor(s): Dilhas; Anna (Basel, CH), Herbert; Mark R (San Diego, CA), Ouerfelli; Ouathek (Fort Lee, NJ), Smith; Nicholas D (San Diego, CA)
Assignee: Aragon Pharmaceuticals, Inc. (San Diego, CA) Sloan-Kettering Institute For Cancer Research (New York, NY)
Application Number:14/406,520
Patent Claim Types:
see list of patent claims
Use; Composition; Compound; Dosage form;

Drugs Protected by US Patent 9,481,663

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate
Janssen Biotech ERLEADA apalutamide TABLET;ORAL 210951-001 Feb 14, 2018 RX Yes Yes   Start Trial   Start Trial Y Y TREATMENT OF NON-METASTATIC, CASTRATION-RESISTANT PROSTATE CANCER (NM-CRPC)   Start Trial
Janssen Biotech ERLEADA apalutamide TABLET;ORAL 210951-001 Feb 14, 2018 RX Yes Yes   Start Trial   Start Trial Y Y TREATMENT OF METASTATIC CASTRATION-SENSITIVE PROSTATE CANCER (MCSPC)   Start Trial
>Applicant >Tradename >Generic Name >Dosage >NDA >Approval Date >TE >Type >RLD >RS >Patent No. >Patent Expiration >Product >Substance >Delist Req. >Patented / Exclusive Use >Submissiondate

Foreign Priority and PCT Information for Patent: 9,481,663

PCT Information
PCT FiledJune 04, 2013PCT Application Number:PCT/US2013/044116
PCT Publication Date:December 12, 2013PCT Publication Number: WO2013/184681

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Serving leading biopharmaceutical companies globally:

Boehringer Ingelheim
Express Scripts

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