Details for Patent: 8,399,450
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Which drugs does patent 8,399,450 protect, and when does it expire?
Patent 8,399,450 protects ZYKADIA and is included in two NDAs.
This patent has one hundred and four patent family members in forty-eight countries.
Summary for Patent: 8,399,450
| Title: | Compounds and compositions as protein kinase inhibitors |
| Abstract: | The invention provides novel pyrimidine and pyridine derivatives and pharmaceutical compositions thereof, and methods for using such compounds. For example, the pyrimidine and pyridine derivatives of the invention may be used to treat, ameliorate or prevent a condition which responds to inhibition of anaplastic lymphoma kinase (ALK) activity, focal adhesion kinase (FAK), zeta-chain-associated protein kinase 70 (ZAP-70), insulin-like growth factor (IGF-1R), or a combination thereof. |
| Inventor(s): | Pierre-Yves Michellys, Wei Pei, Thomas H. Marsilje, Wenshuo Lu, Bei Chen, Tetsuo Uno, Yunho Jin, Tao Jiang |
| Assignee: | Novartis AG |
| Application Number: | US13/172,357 |
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Patent Claim Types: see list of patent claims | Composition; Compound; |
Drugs Protected by US Patent 8,399,450
| Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Submissiondate |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Novartis | ZYKADIA | ceritinib | CAPSULE;ORAL | 205755-001 | Apr 29, 2014 | DISCN | Yes | No | ⤷ Start Trial | ⤷ Start Trial | Y | Y | ⤷ Start Trial | |||
| Novartis | ZYKADIA | ceritinib | TABLET;ORAL | 211225-001 | Mar 18, 2019 | RX | Yes | Yes | ⤷ Start Trial | ⤷ Start Trial | Y | Y | ⤷ Start Trial | |||
| >Applicant | >Tradename | >Generic Name | >Dosage | >NDA | >Approval Date | >TE | >Type | >RLD | >RS | >Patent No. | >Patent Expiration | >Product | >Substance | >Delist Req. | >Patented / Exclusive Use | >Submissiondate |
International Family Members for US Patent 8,399,450
| Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
|---|---|---|---|---|---|
| European Patent Office | 2091918 | ⤷ Start Trial | CA 2015 00047 | Denmark | ⤷ Start Trial |
| European Patent Office | 2091918 | ⤷ Start Trial | C20150037 00157 | Estonia | ⤷ Start Trial |
| European Patent Office | 2091918 | ⤷ Start Trial | 92785 | Luxembourg | ⤷ Start Trial |
| European Patent Office | 2091918 | ⤷ Start Trial | PA2015034 | Lithuania | ⤷ Start Trial |
| >Country | >Patent Number | >Estimated Expiration | >Supplementary Protection Certificate | >SPC Country | >SPC Expiration |
