Details for Patent: 7,772,243
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Which drugs does patent 7,772,243 protect, and when does it expire?
Patent 7,772,243 protects VIZIMPRO and is included in one NDA.
This patent has fifty-six patent family members in forty-six countries.
Summary for Patent: 7,772,243
| Title: | 4-phenylamino-quinazolin-6-yl-amides |
| Abstract: | This invention provides quinazoline compounds of the formula: wherein: R1 is halo; R2 is H or halo; R3 is a) C1-C3 alkyl, optionally substituted by halo; or b) —(CH2)n-morpholino, —(CH2)n-piperidine, —(CH2)n-piperazine, —(CH2)n—-piperazine-N(C1-C3 alkyl), —(CH2)n-pyrrolidine, or —(CH2)n-imidazole; n is 1 to 4; R4 is —(CH2)m-Het; Het is morpholine, piperidine, piperazine, piperazine-N(C1-C3 alkyl), imidazole, pyrrolidine, azepane, 3,4-dihydro-2H-pyridine, or 3,6-dihydro-2H-pyridine, each optionally substituted by alkyl, halo, OH, NH2, NH(C1-C3 alkyl) or N (C1-C3 alkyl)2; m is 1-3; and X is O, S or NH; or a pharmaceutically acceptable salt thereof, as well as processes and intermediate compounds for making them, useful pharmaceutical compositions and methods of using the compounds in the treatment of proliferative diseases. |
| Inventor(s): | Stephen Alan Fakhoury, Helen Tsenwhei Lee, Jessica Elizabeth Reed, Kevin Matthew Schlosser, Karen Elaine Sexton, Haile Tecle, Roy Thomas Winters |
| Assignee: | Warner Lambert Co LLC |
| Application Number: | US11/122,345 |
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Patent Claim Types: see list of patent claims | Composition; Compound; |
| Patent landscape, scope, and claims: |
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Drugs Protected by US Patent 7,772,243
| Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Submissiondate |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Pfizer | VIZIMPRO | dacomitinib | TABLET;ORAL | 211288-001 | Sep 27, 2018 | RX | Yes | No | ⤷ Start Trial | ⤷ Start Trial | Y | Y | ⤷ Start Trial | |||
| Pfizer | VIZIMPRO | dacomitinib | TABLET;ORAL | 211288-002 | Sep 27, 2018 | RX | Yes | No | ⤷ Start Trial | ⤷ Start Trial | Y | Y | ⤷ Start Trial | |||
| Pfizer | VIZIMPRO | dacomitinib | TABLET;ORAL | 211288-003 | Sep 27, 2018 | RX | Yes | Yes | ⤷ Start Trial | ⤷ Start Trial | Y | Y | ⤷ Start Trial | |||
| >Applicant | >Tradename | >Generic Name | >Dosage | >NDA | >Approval Date | >TE | >Type | >RLD | >RS | >Patent No. | >Patent Expiration | >Product | >Substance | >Delist Req. | >Patented / Exclusive Use | >Submissiondate |
International Family Members for US Patent 7,772,243
| Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
|---|---|---|---|---|---|
| European Patent Office | 1746999 | ⤷ Start Trial | 301004 | Netherlands | ⤷ Start Trial |
| European Patent Office | 1746999 | ⤷ Start Trial | PA2019016 | Lithuania | ⤷ Start Trial |
| European Patent Office | 1746999 | ⤷ Start Trial | 122019000080 | Germany | ⤷ Start Trial |
| European Patent Office | 1746999 | ⤷ Start Trial | 2019C/540 | Belgium | ⤷ Start Trial |
| European Patent Office | 1746999 | ⤷ Start Trial | LUC00127 | Luxembourg | ⤷ Start Trial |
| European Patent Office | 1746999 | ⤷ Start Trial | CR 2019 00043 | Denmark | ⤷ Start Trial |
| >Country | >Patent Number | >Estimated Expiration | >Supplementary Protection Certificate | >SPC Country | >SPC Expiration |
