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Details for Patent: 7,750,029
Summary for Patent: 7,750,029
Title: | Remedy for overactive bladder comprising acetic acid anilide derivative as the active ingredient |
Abstract: | (R)-2-(2-aminothiazol-4-yl)-4'-[2-[(2-hydroxy-2-phenylethyl)amino]ethyl]a- cetic acid anilide or its salt shows a potent bladder relaxation effect in "isolated rat bladder smooth muscle relaxation test", dose-dependently lowers the contraction frequency of rhythmic bladder contractions in "rat rhythmic bladder contraction measurement test" and, moreover, prolongs the urination intervals in "urination functions measurement test on cyclophosphamide-induced overactive bladder model rat". Owing to these effects, the above compound is useful as a remedy for ovaractive bladder. |
Inventor(s): | Takasu; Toshiyuki (Tsukuba, JP), Sato; Shuichi (Tsukuba, JP), Ukai; Masashi (Tsukuba, JP), Maruyama; Tatsuya (Tsukuba, JP) |
Assignee: | Astellas Pharma Inc. (Tokyo, JP) |
Application Number: | 10/534,290 |
Patent Claim Types: see list of patent claims | Use; |
Drugs Protected by US Patent 7,750,029
Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Patent Submitted |
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Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Patent Submitted |
Foreign Priority and PCT Information for Patent: 7,750,029
Foriegn Application Priority Data | ||
Foreign Country | Foreign Patent Number | Foreign Patent Date |
Japan | 2002-323792 | Nov 07, 2002 |
PCT Information | |||
PCT Filed | November 04, 2003 | PCT Application Number: | PCT/JP03/14065 |
PCT Publication Date: | May 21, 2004 | PCT Publication Number: | WO2004/041276 |
International Patents Family Members for US Patent 7,750,029
Country | Document Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
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Austria | 500827 | ➤ Sign Up | |||
Australia | 2003284700 | ➤ Sign Up | |||
Brazil | 0316080 | ➤ Sign Up | |||
Canada | 2503570 | ➤ Sign Up | |||
Country | Document Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |