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Generated: May 26, 2019

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Details for Patent: 7,417,042

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Which drugs does patent 7,417,042 protect, and when does it expire?

Patent 7,417,042 protects KYPROLIS and is included in one NDA.

This patent has eighty-four patent family members in twenty-six countries.

Summary for Patent: 7,417,042
Title:Compounds for enzyme inhibition
Abstract: Peptide-based compounds including heteroatom-containing, three-membered rings efficiently and selectively inhibit specific activities of N-terminal nucleophile (Ntn) hydrolases. The activities of those Ntn having multiple activities can be differentially inhibited by the compounds described. For example, the chymotrypsin-like activity of the 20S proteasome may be selectively inhibited with the inventive compounds. The peptide-based compounds include an epoxide or aziridine, and functionalization at the N-terminus. Among other therapeutic utilities, the peptide-based compounds are expected to display anti-inflammatory properties and inhibition of cell proliferation.
Inventor(s): Smyth; Mark S. (Foster City, CA), Laidig; Guy J. (Menlo Park, CA)
Assignee: Proteolix, Inc. (South San Francisco, CA)
Application Number:11/199,899
Patent Litigation and PTAB cases: See patent lawsuits and PTAB cases for patent 7,417,042
Prior Art and Litigation SupportOrder Prior Art and Litigation support for Patent 7,417,042
Patent Claim Types:
see list of patent claims
Compound; Composition;

Drugs Protected by US Patent 7,417,042

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate
Onyx Therap KYPROLIS carfilzomib POWDER;INTRAVENOUS 202714-003 Jun 7, 2018 RX Yes No ➤ Sign Up ➤ Sign Up Y Y ➤ Sign Up
Onyx Therap KYPROLIS carfilzomib POWDER;INTRAVENOUS 202714-002 Jun 3, 2016 RX Yes No ➤ Sign Up ➤ Sign Up Y Y ➤ Sign Up
Onyx Therap KYPROLIS carfilzomib POWDER;INTRAVENOUS 202714-001 Jul 20, 2012 RX Yes Yes ➤ Sign Up ➤ Sign Up Y Y ➤ Sign Up
Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate

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International Family Members for US Patent 7,417,042

Country Patent Number Estimated Expiration Supplementary Protection Certificate SPC Country SPC Expiration
Austria 494298 ➤ Sign Up
Austria 496062 ➤ Sign Up
Australia 2005238445 ➤ Sign Up
Australia 2005271232 ➤ Sign Up
Australia 2005295183 ➤ Sign Up
Australia 2012203602 ➤ Sign Up
Country Patent Number Estimated Expiration Supplementary Protection Certificate SPC Country SPC Expiration

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Serving hundreds of leading biopharmaceutical companies globally:

Federal Trade Commission
UBS
Boehringer Ingelheim
Merck
Harvard Business School
Queensland Health

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