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Last Updated: April 20, 2024

Details for Patent: 7,205,302


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Which drugs does patent 7,205,302 protect, and when does it expire?

Patent 7,205,302 protects UPTRAVI and is included in two NDAs.

This patent has twenty-one patent family members in sixteen countries.

Summary for Patent: 7,205,302
Title:Heterocyclic compound derivatives and medicines
Abstract: The present invention provides a compound which is useful as a PGI.sub.2 receptor agonist, and a pharmaceutical composition. The present invention is directed to a pharmaceutical composition comprising a compound represented by the following formula [1]: ##STR00001## (R.sup.1 and R.sup.2 are the same or different and each represents optionally substituted aryl, Y represents N or CH, Z represents N or CH, A represents NH, NR.sup.5, O, S, or ethylene, R.sup.5 represents alkyl, D represents alkylene or alkenylene, E represents phenylene or single bond, G represents O, S, or CH.sub.2, R.sup.3 and R.sup.4 are the same or different and each represents hydrogen or alkyl, Q represents carboxy, alkoxycarbonyl, tetrazolyl, carbamoyl, or N-(alkylsulfonyl)carbamoyl), or a pharmaceutically acceptable salt thereof as an active ingredient.
Inventor(s): Asaki; Tetsuo (Kyoto, JP), Hamamoto; Taisuke (Osaka, JP), Kuwano; Keiichi (Osaka, JP)
Assignee: Nippon Shinyaku Co., Ltd. (Kyoto, JP)
Application Number:10/476,196
Patent Litigation and PTAB cases: See patent lawsuits and PTAB cases for patent 7,205,302
Patent Claim Types:
see list of patent claims
Composition; Compound; Use;

Drugs Protected by US Patent 7,205,302

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate
Actelion UPTRAVI selexipag POWDER;INTRAVENOUS 214275-001 Jul 29, 2021 RX Yes Yes ⤷  Try a Trial ⤷  Try a Trial Y Y METHOD OF TREATING PULMONARY ARTERIAL HYPERTENSION COMPRISING ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG ⤷  Try a Trial
Actelion UPTRAVI selexipag TABLET;ORAL 207947-001 Dec 21, 2015 AB RX Yes No ⤷  Try a Trial ⤷  Try a Trial Y Y METHOD OF TREATING PULMONARY ARTERIAL HYPERTENSION COMPRISING ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG ⤷  Try a Trial
Actelion UPTRAVI selexipag TABLET;ORAL 207947-002 Dec 21, 2015 AB RX Yes Yes ⤷  Try a Trial ⤷  Try a Trial Y Y METHOD OF TREATING PULMONARY ARTERIAL HYPERTENSION COMPRISING ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG ⤷  Try a Trial
Actelion UPTRAVI selexipag TABLET;ORAL 207947-003 Dec 21, 2015 AB RX Yes No ⤷  Try a Trial ⤷  Try a Trial Y Y METHOD OF TREATING PULMONARY ARTERIAL HYPERTENSION COMPRISING ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG ⤷  Try a Trial
Actelion UPTRAVI selexipag TABLET;ORAL 207947-004 Dec 21, 2015 AB RX Yes No ⤷  Try a Trial ⤷  Try a Trial Y Y METHOD OF TREATING PULMONARY ARTERIAL HYPERTENSION COMPRISING ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG ⤷  Try a Trial
Actelion UPTRAVI selexipag TABLET;ORAL 207947-005 Dec 21, 2015 RX Yes No ⤷  Try a Trial ⤷  Try a Trial Y Y METHOD OF TREATING PULMONARY ARTERIAL HYPERTENSION COMPRISING ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG ⤷  Try a Trial
Actelion UPTRAVI selexipag TABLET;ORAL 207947-006 Dec 21, 2015 RX Yes No ⤷  Try a Trial ⤷  Try a Trial Y Y METHOD OF TREATING PULMONARY ARTERIAL HYPERTENSION COMPRISING ADMINISTERING A PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG ⤷  Try a Trial
>Applicant >Tradename >Generic Name >Dosage >NDA >Approval Date >TE >Type >RLD >RS >Patent No. >Patent Expiration >Product >Substance >Delist Req. >Patented / Exclusive Use >Submissiondate

Foreign Priority and PCT Information for Patent: 7,205,302

Foriegn Application Priority Data
Foreign Country Foreign Patent Number Foreign Patent Date
Japan2001-129765Apr 26, 2001
PCT Information
PCT FiledApril 25, 2002PCT Application Number:PCT/JP02/04118
PCT Publication Date:November 07, 2002PCT Publication Number: WO02/088084

International Family Members for US Patent 7,205,302

Country Patent Number Estimated Expiration Supplementary Protection Certificate SPC Country SPC Expiration
Brazil 0209249 ⤷  Try a Trial
Brazil PI0209249 ⤷  Try a Trial
Canada 2445344 ⤷  Try a Trial
China 1301973 ⤷  Try a Trial
China 1516690 ⤷  Try a Trial
Germany 60217674 ⤷  Try a Trial
Denmark 1400518 ⤷  Try a Trial
>Country >Patent Number >Estimated Expiration >Supplementary Protection Certificate >SPC Country >SPC Expiration

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