Details for Patent: 5,610,163
Summary for Patent: 5,610,163
| Title: | Esters of thienyl carboxylic acids and amino alcohols and their quaternization products |
| Abstract: | Compounds of the formula ##STR1## of which, in exemplary compounds, the thienyl group is attached via the 2-position and:(a) A is 3α-(6β, 7β-epoxy)-tropanyl methobromide and R1 is 2-thienyl;(b) A is 3α-(6, 7dehydro)-tropanyl methobromide and R1 is 2-thienyl;(c) A is 3β-tropanyl methobromide and R1 is 2-thienyl; and,(d) A is 3α-(N-isopropyl)-nortropanyl methobromide and R1 is cyclopentyl.These are anticholinergics. Administered by inhalation, they are useful for the treatment of chronic obstructive bronchitis or slight to moderately severe asthma. Administered by the intravenous or oral routes, they are useful for the treatment of vagally induced sinus bradycardia. |
| Inventor(s): | Rolf Banholzer, Rudolf Bauer, Richard Reichl |
| Assignee: | Boehringer Ingelheim GmbH |
| Application Number: | US08/405,111 |
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Patent Claim Types: see list of patent claims | Use; Composition; Dosage form; |
Drugs Protected by US Patent 5,610,163
| Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Submissiondate |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| >Applicant | >Tradename | >Generic Name | >Dosage | >NDA | >Approval Date | >TE | >Type | >RLD | >RS | >Patent No. | >Patent Expiration | >Product | >Substance | >Delist Req. | >Patented / Exclusive Use | >Submissiondate |
Foreign Priority and PCT Information for Patent: 5,610,163
| Foriegn Application Priority Data | ||
| Foreign Country | Foreign Patent Number | Foreign Patent Date |
| Germany | 39 31 041.8 | Sep 16, 1989 |
International Family Members for US Patent 5,610,163
| Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
|---|---|---|---|---|---|
| European Patent Office | 0418716 | ⤷ Start Trial | SPC/GB02/036 | United Kingdom | ⤷ Start Trial |
| European Patent Office | 0418716 | ⤷ Start Trial | 05C0039 | France | ⤷ Start Trial |
| European Patent Office | 0418716 | ⤷ Start Trial | C300084 | Netherlands | ⤷ Start Trial |
| European Patent Office | 0418716 | ⤷ Start Trial | 0290010-8 | Sweden | ⤷ Start Trial |
| European Patent Office | 0418716 | ⤷ Start Trial | 300084 | Netherlands | ⤷ Start Trial |
| >Country | >Patent Number | >Estimated Expiration | >Supplementary Protection Certificate | >SPC Country | >SPC Expiration |
