Details for Patent: 4,011,258
Summary for Patent: 4,011,258
| Title: | Orally active bronchospasmolytic compounds |
| Abstract: | Novel compounds are disclosed having useful activity as bronchodilators of improved longevity of action and reduced incidence of side effects. These compounds are described by the formula: ##STR1## wherein R1 is a member of the class consisting of tertiary butyl and cyclobutyl, and R2 is a hydrogen or 2 to 5 carbon atom acyl radical, and pharmaceutically acceptable salts thereof. The activity of these compounds is compared to previously known bronchodilators such as 1-(3', 5'-dihydroxyphenyl)-2-(isopropylamino)-ethanol, having the common name orciprenaline, and 1-(3', 4'-dihydroxyphenyl-2-isopropylamino-ethanol, having the common name isoprenaline. |
| Inventor(s): | Kjell Ingvar Leopold Wetterlin, Leif Ake Svensson |
| Assignee: | Draco AB |
| Application Number: | US05/593,424 |
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Patent Claim Types: see list of patent claims | Compound; |
Drugs Protected by US Patent 4,011,258
| Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Submissiondate |
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International Family Members for US Patent 4,011,258
| Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
|---|---|---|---|---|---|
| Austria | 286964 | ⤷ Start Trial | |||
| Austria | 287678 | ⤷ Start Trial | |||
| Austria | 287679 | ⤷ Start Trial | |||
| Austria | 288356 | ⤷ Start Trial | |||
| Belgium | 704932 | ⤷ Start Trial | |||
| Switzerland | 510625 | ⤷ Start Trial | |||
| >Country | >Patent Number | >Estimated Expiration | >Supplementary Protection Certificate | >SPC Country | >SPC Expiration |
