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Details for Patent: 3,978,121
Title: | 5H Dibenzo[a,d]cycloheptene derivatives |
Abstract: | Compounds of 5H dibenzo[a,d]-cycloheptenes and 10,11-dihydro-5H-dibenzo[a,d]cycloheptenes which are substituted at their 5-carbon atom with an N-cyanoaminopropyl or an N-cyanoaminopropylidene radical. |
Inventor(s): | Engelhardt; Edward L. (Gwynedd Valley, PA) |
Assignee: | Merck & Co., Inc. (Rahway, NJ) |
Filing Date: | Apr 11, 1975 |
Application Number: | 05/567,165 |
Claims: | 1. A compound selected from the group consisting of: ##SPC10## wherein R is a lower alkyl radical, Y is selected from the group consisting of hydrogen and halogen and X and X' are selected from the group consisting of hydrogen, an alkyl group having up to 6 carbon atoms, an alkenyl group having up to 6 carbon atoms, a perfluoroalkyl group having up to 4 carbon atoms, phenyl, an acyl group having up to 4 carbon atoms, a perfluoroacyl group having up to 4 carbon atoms, amino, an alkylamino group having up to 4 carbon atoms, a dialkylamino group having up to 8 carbon atoms, an acylamino group having up to 4 carbon atoms, a perfluoroacylamino group having up to 4 carbon atoms, an alkylsulfonylamino group having up to 4 carbon atoms, halogen, hydroxyl, an alkoxyl group having up to 4 carbon atoms, a perfluoroalkoxyl group having up to 4 carbon atoms, cyano carboxy, carbenyl, an alkylcarbamyl group having up to 5 carbon atoms, a dialkylcarbamyl group having up to 9 carbon atoms, a carbalkoxy group having up to 6 carbon atoms, mercapto, an alkylmercapto group having up to 4 carbon atoms, a perfluoroalkylmercapto group having up to 4 carbon atoms, an alkylsulfonyl group having up to 4 carbon atoms, a perfluoroalkylsulfonyl group having up to 4 carbon atoms, sulfamoyl, an alkylsulfamoyl group having up to 4 carbon atoms and a dialkylsulfamoyl group having up to 8 carbon atoms. 2. A 5-(3-N-cyano-N-lower alkylaminopropylidene)-5H-dibenzo[a,d]cycloheptene. 3. A 5-(3-N-cyano-N-lower alkylaminopropylidene)-10,11-dihydro-5H-dibenzo[a,d]cycloheptene. 4. A 5-(3-N-cyano-N-lower alkylaminopropyl)-5H-dibenzo[a,d]cycloheptene. 5. A 5-(3-N-cyano-N-lower alkylaminopropyl)-10,11-dihydro-5H-dibenzo[a,d]cycloheptene. 6. 5-(3-N-Cyano-N-methylaminopropyl)-5H-dibenzo-[a,d]cycloheptene. 7. 5-(3-N-Cyano-N-methylaminopropylidene)-10,11-dihydro-5H-dibenzo [a,d]cycloheptene. |