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Details for Patent: 3,885,037

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Details for Patent: 3,885,037

Title: Method of producing anorexia using imidazolinyl phenyl carbonyl compounds, their acid addition salts and related compounds
Abstract:This invention is concerned with tetrahydropyrimidinyl phenyl carbonyl acid addition salts, imidazolinyl phenyl carbonyl acid addition salts, dihydroimidazoisoindolols, tetrahydropyrimidoisoindolols, and tetrahydropyrimidoisoindolol acid addition salts which are all pharmacologically efficacious as anti-depressants. The tetrahydropyrimidinyl phenyl carbonyl acid addition salts, the tetrahydropyrimidoisoindolols and the tetrahydropyrimidoisoindolol acid addition salts are also efficacious as diuretics while the imidazolinyl phenyl carbonyl acid addition salts and the dihydroimidazoisoindolols are efficacious as anorexiants. This invention is also concerned with several processes for the preparation of these compounds.
Inventor(s): Sulkowski; Theodore S. (Wayne, PA)
Assignee: American Home Products Corporation (New York, NY)
Filing Date:Sep 06, 1973
Application Number:05/394,952
Claims:1. A method of producing anorexia in an animal in need thereof which comprises administering to said animal an effective amount of a compound having the formula ##SPC7##

wherein R.sub.2 is selected from the group consisting of hydrogen, halogen, amino, lower alkylamino, lower alkyl, and lower alkoxy; R.sub.3 is hydrogen when R.sub.2 and R.sub.3 are dissimilar and when R.sub.2 and R.sub.3 are the same they are both selected from the group consisting of hydrogen, halogen, lower alkyl, and lower alkoxy; and R.sub.4 is selected from the group consisting of phenyl, monohalophenyl, dihalogphenyl, mono(lower)alkylphenyl, di(lower)alkylphenyl, trifluoromethylphenyl, mono(lower)alkoxy phenyl, and di(lower)alkoxyphenyl.

2. A method of producing anorexia in an animal in need thereof which comprises administering to said animal an effective amount of a compound having the formula ##SPC8##

wherein R.sub.2 is selected from the group consisting of hydrogen, halogen, amino, lower alkylamino, lower alkyl, and lower alkoxy; R.sub.3 is hydrogen when R.sub.2 and R.sub.3 are dissimilar and when R.sub.2 and R.sub.3 are the same they are both selected from the group consisting of hydrogen, halogen, lower alkyl, and lower alkoxy; R.sub.1 is selected from the group consisting of phenyl, monohalophenyl, dihalophenyl, mono(lower)alkylphenyl, di(lower)alkylphenyl, trifluoromethylphenyl, mono(lower)alkoxyphenyl, and di(lower)alkoxyphenyl; and HA is a pharmaceutically acceptable acid.
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