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Last Updated: December 2, 2021

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Patent: 9,663,523

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Summary for Patent: 9,663,523
Title:BET protein-inhibiting 5-aryltriazoleazepines
Abstract: The present invention relates to BET-protein-inhibitory, in particular BRD4-inhibitory 5-aryltriazoloazepines of the general formula (I) ##STR00001## in which R.sup.1, R.sup.2, R.sup.3 and R.sup.4 have the meanings given for the general formula (I), to pharmaceutical compositions comprising the compounds according to the invention, and to the prophylactic and therapeutic use thereof for hyperproliferative disorders, especially for neoplastic disorders. The present invention further relates to the use of BET protein inhibitors in viral infections, in neurodegenerative disorders, in inflammatory diseases, in atherosclerotic disorders and in male fertility control.
Inventor(s): Schmees; Norbert (Berlin, DE), Kuhnke; Joachim (Potsdam, DE), Haendler; Bernard (Berlin, DE), Neuhaus; Roland (Berlin, DE), Lejeune; Pascale (Berlin, DE), Siegel; Stephan (Berlin, DE), Kruger; Martin (Berlin, DE), Fernandez-Montalvan; Amaury Ernesto (Berlin, DE), Kunzer; Hermann (Berlin, DE), Gallenkamp; Daniel (Wuppertal, DE)
Assignee: BAYER PHARMA AKTIENGESELLSCHAFT (Berlin, DE)
Application Number:14/432,158
Patent Claims:see list of patent claims

Details for Patent 9,663,523

Applicant Tradename Biologic Ingredient Dosage Form BLA Approval Date Patent No. Expiredate
Recordati Rare Diseases, Inc. ELSPAR asparaginase For Injection 101063 1978-01-10 ⤷  Free Forever Trial 2032-09-28
Genentech, Inc. RITUXAN rituximab Injection 103705 1997-11-26 ⤷  Free Forever Trial 2032-09-28
Idec Pharmaceuticals Corp. RITUXAN rituximab Injection 103737 2002-02-19 ⤷  Free Forever Trial 2032-09-28
Genentech, Inc. HERCEPTIN trastuzumab For Injection 103792 1998-09-25 ⤷  Free Forever Trial 2032-09-28
Genentech, Inc. HERCEPTIN trastuzumab For Injection 103792 2017-02-10 ⤷  Free Forever Trial 2032-09-28
Eli Lilly And Company ERBITUX cetuximab Injection 125084 2004-02-12 ⤷  Free Forever Trial 2032-09-28
>Applicant >Tradename >Biologic Ingredient >Dosage Form >BLA >Approval Date >Patent No. >Expiredate

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Johnson and Johnson
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McKinsey

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