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Patent: 5,585,397

Summary for Patent: 5,585,397

Title: Sulfonamide inhibitors of aspartyl protease
Abstract:The present invention relates to a novel class of sulfonamides which are aspartyl protease inhibitors. In one embodiment, this invention relates to a novel class of HIV aspartyl protease inhibitors characterized by specific structural and physicochemical features. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibiting HIV-1 and HIV-2 protease activity and consequently, may be advantageously used as anti-viral agents against the HIV-1 and HIV-2 viruses. This invention also relates to methods for inhibiting the activity of HIV aspartyl protease using the compounds of this invention and methods for screening compounds for anti-HIV activity.
Inventor(s): Tung; Roger D. (Arlington, MA), Murcko; Mark A. (Holliston, MA), Bhisetti; Govinda R. (Lexington, MA)
Assignee: Vertex Pharmaceuticals, Incorporated (Cambridge, MA)
Application Number:08/142,327
Patent Claim Types:
see list of patent claims
Compound; Composition;
Patent PDF download available with subscription

Glossary
Applicant Tradename Generic Name Dosage NDA Approval Date Type RLD Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use
Glaxosmithkline
AGENERASE
amprenavir
CAPSULE;ORAL021007Apr 15, 1999DISCNNo5,585,397<disabled>
Glaxosmithkline
AGENERASE
amprenavir
SOLUTION;ORAL021039Apr 15, 1999DISCNNo5,585,397<disabled>
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Foreign Priority and PCT Information for Patent: 5,585,397

PCT Information
PCT FiledSeptember 07, 1993PCT Application Number:PCT/US93/08458
PCT Publication Date:March 17, 1994PCT Publication Number: WO94/05639

International Patent Family for Patent: 5,585,397

Country Document Number Publication Date
ARIPO950Mar 28, 2001
ARIPO9701119Oct 31, 1997
ARIPO390Aug 02, 1995
ARIPO9300572Oct 31, 1993
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